Skip to main content

In Search of The Perfect Sleep Aid

 For many years, modern medicine has been searching for the perfect sleeping pills. Sleeping pills are a special topic in medicine because they have a lot to do with addiction medicine. Of course, not every sleeping pill can cause addiction, but lighter sleeping pills such as valerian tablets, doxylamine succinate (contained in Schlafsterne), melatonin (or Circadin) have short and insufficient effects.


Benzodiazepines, on the other hand, relieve anxiety, which often leads to sleep disorders and are often used by GPs as sleeping pills, although this is not correct. Antidepressants such as mirtazapine are more often used as sleeping pills, but patients often complain of fatigue and drowsiness after their use, which is incompatible with driving, for example.


Z-drugs are the 3rd choice of sleep medicine, they have a long and sufficient effect, but can be very addictive. There are patients who struggle for years with addiction to zolpidem, or zopiclone. Many GPs give up in this fight and prescribe these drugs simply because the patients are already addicted.


Benzodiazepines and Z-drugs have a clear withdrawal reaction even when used briefly.


But we are not giving up.



It has long been known that H1 inhibitors of first (such as clemastine) and second generation (such as cetirizine), which are used as anti-allergic agents without hesitation, have a strong drowsiness effect and even severe sleepiness as a side effect. This drowsiness can last up to 12 hours (perfect nap, right?).


Can we use side effects as the main effect? - Why not? The only “downside” is that we are also treating an allergy predisposition in this case.


The only side effect of antihistamines is mild dry mouth, which is temporary. Antihistamines can also be used without hesitation when withdrawal effects of benzodiazepines occur.


Antihistamines are inexpensive.


Of course, the question is who will do the clinical trial and give us the final answer. 


Translated with DeepL.com (free version)

Comments

Popular posts from this blog

Why Ozempic Causes Blindness?

What Is Ozempic? Ozempic (semaglutide) Injection is a  glucagon -like  peptide  1 (GLP-1) receptor  agonist  indicated as an adjunct to diet and exercise to improve glycemic control in adults with type 2  diabetes mellitus . What Are Side Effects of Ozempic? Ozempic may cause serious side effects including: a lump in the neck, difficulty swallowing, cough, shortness of breath, difficulty breathing, upper abdominal pain, nausea, vomiting, blurred vision, spots or dark strings floating in your vision, fluctuating vision, vision loss, dark or empty areas in your vision, shakiness, nervousness, anxiety, sweating, chills, clamminess, irritability, impatience, confusion, fast heartrate, lightheadedness , dizziness, hunger, decreased urination, swelling in your legs, ankles, or feet, fatigue, rash, itching, and shock Get medical help right away, if you have any of the symptoms listed above....

New Look on Antihypertensive Therapy

  Angiotensin converting enzyme 2   Angiotensin converting enzyme 2, or ACE2, is an exopeptidase expressed primarily by vascular endothelial cells in the heart and kidneys, but also in respiratory epithelia[1] and in the gastrointestinal tract. It is the target of several coronaviruses, including SARS-CoV and SARS-CoV-2. 2 Biochemistry ACE2 is a transmembrane metallocarboxypeptidase composed of 805 amino acids. Zinc and chloride ions act as cofactors. The extracellular region consists of two domains, a zinc metallopeptidase domain and a C-terminal collectrin homology domain. The enzyme exhibits homology to angiotensin converting enzyme (ACE). ACE2 is encoded by the ACE2 gene on the X chromosome (gene locus Xp22.2). In addition to being expressed as a transmembrane protein, a soluble form exists in serum. 3 Function ACE2 cleaves angiotensin II into angiotensin (1-7), which has anti-inflammatory and lung protective effects via MAS and AT2 receptors. 4 Clinical ...